Bringing Assays and Automation Together for Lower Throughput Kinase Profiling

Kinase profiling during drug discovery is a necessary process to confirm inhibitor selectivity and assess off-target activity. While automation is necessary to screen and identify putative inhibitors, it can also provide benefit for follow-up characterization studies where throughput is not a primary concern. This scientific poster presents a semi-automated workflow for lower throughput kinase profiling applications.